Drug Classifications

Major drug classes with generic name suffixes, mechanisms of action, common side effects, and nursing implications.

Drug Classification Quick Reference

Recognizing drug suffixes helps identify the class, mechanism, and expected side effects of unfamiliar medications.

Cardiovascular Medications

ClassSuffix/ExamplesMechanism of ActionKey Side EffectsNursing Implications
ACE Inhibitors-pril (lisinopril, enalapril, captopril, ramipril)Block conversion of angiotensin I to II; reduce preload/afterloadDry cough (most common), hyperkalemia, angioedema (rare but serious), hypotensionMonitor K+ and renal function; hold for hyperkalemia; contraindicated in pregnancy; report persistent cough
ARBs-sartan (losartan, valsartan, irbesartan)Block angiotensin II receptors; similar effect to ACE inhibitorsHyperkalemia, hypotension, dizzinessAlternative if ACE inhibitor cough; still monitor K+ and BUN/Cr; contraindicated in pregnancy
Beta-Blockers-olol (metoprolol, atenolol, propranolol, carvedilol)Block beta-adrenergic receptors; decrease HR, BP, myocardial O2 demandBradycardia, hypotension, fatigue, bronchospasm, masks hypoglycemiaHold if HR < 60 or SBP < 90; do NOT stop abruptly; avoid in asthma (non-selective); monitor glucose in diabetics
Calcium Channel Blockers-dipine (amlodipine, nifedipine) and diltiazem, verapamilBlock calcium entry into vascular smooth muscle and cardiac cells; vasodilationPeripheral edema, constipation (verapamil), headache, dizziness, bradycardiaMonitor HR and BP; avoid grapefruit juice; assess for peripheral edema
Statins-statin (atorvastatin, simvastatin, rosuvastatin, pravastatin)Inhibit HMG-CoA reductase; lower LDL cholesterolMyalgia/myopathy (report muscle pain), rhabdomyolysis (rare), hepatotoxicityMonitor LFTs, CK if muscle complaints; take in evening (most production at night); avoid grapefruit with some statins
AnticoagulantsHeparin, enoxaparin (-parin), warfarin, rivaroxaban (-xaban), apixaban, dabigatranPrevent clot formation through various pathwaysBleeding (all); HIT (heparin); see medication cheat sheetMonitor aPTT (heparin), INR (warfarin); teach bleeding precautions; DOACs have fewer monitoring requirements
Loop Diuretics-semide (furosemide/Lasix, bumetanide)Block Na/K/Cl transport in Loop of Henle; potent diuresisHypokalemia, hyponatremia, hypotension, ototoxicity, dehydrationMonitor K+ (supplement PRN); I&O, daily weights; give in AM to prevent nocturia; monitor hearing
Thiazide Diuretics-thiazide (hydrochlorothiazide, chlorthalidone)Inhibit Na reabsorption in distal tubuleHypokalemia, hyperglycemia, hyperuricemia, hypercalcemiaMonitor electrolytes; may worsen gout; mild diuretic; often combined with other antihypertensives
K-Sparing DiureticsSpironolactone, triamterene, amilorideBlock aldosterone or Na channels in collecting duct; retain KHyperkalemia, gynecomastia (spironolactone)Do NOT give with K supplements or ACE inhibitors/ARBs without close monitoring; monitor K+

CNS Medications

ClassSuffix/ExamplesMOAKey Side EffectsNursing Implications
Benzodiazepines-pam, -lam (diazepam, lorazepam, midazolam, alprazolam)Enhance GABA activity; CNS depressionSedation, respiratory depression, dependence, paradoxical excitation (elderly)Antidote: flumazenil; avoid alcohol; fall precautions; taper to discontinue; short-term use preferred
Opioid Analgesics-one, -ine, -ol (morphine, hydrocodone, oxycodone, fentanyl, codeine)Bind opioid receptors; pain relief, CNS depressionRespiratory depression, constipation, sedation, nausea, urinary retention, hypotensionAntidote: naloxone (Narcan); assess RR before giving (hold if < 12); bowel regimen; assess pain scale; monitor sedation level
AnticonvulsantsPhenytoin (Dilantin), levetiracetam, valproic acid, carbamazepineStabilize neuronal membranes; reduce seizure activityVary by drug: gingival hyperplasia (phenytoin), hepatotoxicity (valproic acid), Stevens-Johnson (lamotrigine, carbamazepine)Monitor therapeutic levels; phenytoin: IV rate ≤ 50 mg/min (cardiac monitoring); never mix with dextrose; oral care for gingival hyperplasia

Anti-Infective Medications

ClassSuffix/ExamplesKey Considerations
Penicillins-cillin (amoxicillin, ampicillin, piperacillin)Ask about allergy (cross-reactivity with cephalosporins ~1–2%); take full course; monitor for anaphylaxis
Cephalosporinscef-, ceph- (cephalexin, ceftriaxone, cefazolin)Cross-allergy with penicillin possible; avoid alcohol with some (disulfiram-like reaction); monitor renal function
Fluoroquinolones-floxacin (ciprofloxacin, levofloxacin, moxifloxacin)Risk of tendon rupture (especially Achilles); avoid in children < 18; photosensitivity; do not take with antacids, dairy, or iron (chelation)
Aminoglycosides-mycin, -micin (gentamicin, tobramycin, amikacin)Ototoxicity (hearing loss, tinnitus) and nephrotoxicity; monitor peak/trough levels, BUN/Cr, hearing; adequate hydration
Macrolides-thromycin (azithromycin, erythromycin, clarithromycin)GI upset common; QT prolongation risk; many drug interactions (CYP3A4); alternative for penicillin allergy
VancomycinVancomycinTrough level: 15–20 mcg/mL; Red Man Syndrome (histamine reaction — slow infusion over 60+ min); ototoxic, nephrotoxic; monitor levels, renal function

Endocrine Medications

ClassExamplesKey Nursing Points
BiguanidesMetformin (Glucophage)First-line for Type 2 DM; hold 48 hrs before/after contrast dye; risk of lactic acidosis; do not use in renal impairment; GI side effects common
Sulfonylureas-ide (glipizide, glyburide, glimepiride)Stimulate insulin secretion; risk of hypoglycemia; take 30 min before meals; weight gain
Corticosteroids-sone, -olone (prednisone, prednisolone, methylprednisolone, dexamethasone, hydrocortisone)Never stop abruptly (adrenal crisis); immunosuppression; hyperglycemia; osteoporosis; GI irritation; Cushing features with long-term use; take with food; give in AM to mimic natural cortisol
Thyroid HormonesLevothyroxine (Synthroid)Take on empty stomach, 30–60 min before breakfast; lifelong therapy for hypothyroidism; monitor TSH; separate from calcium, iron, antacids by 4 hours

Suffix Quick Reference

SuffixDrug Class
-prilACE Inhibitors
-sartanARBs
-ololBeta-Blockers
-dipineCalcium Channel Blockers (dihydropyridine)
-statinHMG-CoA Reductase Inhibitors
-pam / -lamBenzodiazepines
-prazoleProton Pump Inhibitors
-tidineH2 Receptor Blockers
-cillinPenicillins
-floxacinFluoroquinolones
-mycin / -micinAminoglycosides
-thromycinMacrolides
-cyclineTetracyclines
-mabMonoclonal Antibodies
-nibKinase Inhibitors
-sone / -oloneCorticosteroids
-xabanFactor Xa Inhibitors (DOACs)
-parinHeparins (LMWH)
-setron5-HT3 Antagonists (antiemetics)
-triptanSerotonin Agonists (migraine)
-gliptinDPP-4 Inhibitors (diabetes)
-glutideGLP-1 Receptor Agonists (diabetes/weight loss)
-gliflozinSGLT2 Inhibitors (diabetes)